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LGD-4033 (Ligandrol)

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Description

Description

Sample size: 50ml  |  10mg/ml  |   500mg  |   99% Purity

M.Wt: 338.25
Formula: C14H12F6N2O – 4-((R)-2-((R)-2,2,2-trifluoro-1-hydroxyethyl)pyrrolidin-1-yl)-2-trifluoroMethyl)benzonitrile
Solubility: DMSO
Purity: >99%
Storage: at 20℃ 2 years
Half life: 24 hours
CAS No.: 1165910-22-4

 

Activity of LGD-4033:

LGD-4033 is a selective androgen receptor modulator a novel non-steroidal, oral SARM that binds to AR with high affinity (Ki of ~1 nM) and selectivity, class of androgen receptor (AR) ligands that is tissue selective, developed to treat muscle wasting associated with cancer, acute and chronic illness and age-related muscle loss. Expected to produce the therapeutic benefits of testosterone with improved safety, tolerability and patient acceptance due to tissue-selective mechanism of action and an oral route of administration. It demonstrates anabolic activity in muscles, anti-resorptive and anabolic activity in bones and a robust selectivity for muscle and bone versus prostate and sebaceous glands. LGD-4033 has recently completed a Phase I Multiple Ascending Dose study in healthy volunteers this randomized, double-blind, placebo-controlled Phase I study established the safety and tolerability up to doses of 22 mg.[1] [2] [3] [4]

*This article is intended for educational / informational purposes only. THIS PRODUCT IS INTENDED AS A RESEARCH CHEMICAL ONLY. This designation allows the use of research chemicals strictly for in vitro testing and laboratory experimentation only.
 

For bulk purchases, please contact quant@researchsarms.co.uk

For Custom soloution orders, please contact custom@researchsarms.co.uk

Store at room temperature out of direct light.

This product is for research only and not for consumption.

1ML applicator is included with each order for your convenience but more can be added to your shopping cart.

Testing Documentation
Full Testing documentation will be uploaded to individual pages soon. To request it proir to this please email us at info@researchsarms.co.uk
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